CAS 360791-49-7 4BP-TQS - Analytical Products / Alfa Chemistry

CAT	AP360791497
CAS	360791-49-7
MDL Number	MFCD00981752
Molecular Weight	405.31
InChI Key	YNCXHXYZTLIZTO-UHFFFAOYSA-N

Description	≥98% (HPLC)
Solubility	DMSO: 20 mg/mL, clear
Assay	≥98% (HPLC)
Color	white to beige
Form	powder
Size	5MG, 25MG
Storage Conditions	−20°C

1

A Series of α7 Nicotinic Acetylcholine Receptor Allosteric Modulators With Close Chemical Similarity but Diverse Pharmacological Properties

JasKiran K Gill, Persis Dhankher, Tom D Sheppard, Emanuele Sher, Neil S Millar

Mol Pharmacol. 2012 May;81(5):710-8.

PMID: 22328718

1

Activation of α7 Nicotinic Receptors by Orthosteric and Allosteric Agonists: Influence on Single-Channel Kinetics and Conductance

Magda M Pałczyńska, Marie Jindrichova, Alasdair J Gibb, Neil S Millar

Mol Pharmacol. 2012 Nov;82(5):910-7.

PMID: 22874415

1

Agonist Activation of alpha7 Nicotinic Acetylcholine Receptors via an Allosteric Transmembrane Site

Jaskiran K Gill, Mari Savolainen, Gareth T Young, Ruud Zwart, Emanuele Sher, Neil S Millar

Proc Natl Acad Sci U S A. 2011 Apr 5;108(14):5867-72.

PMID: 21436053

1

Contrasting Properties of α7-selective Orthosteric and Allosteric Agonists Examined on Native Nicotinic Acetylcholine Receptors

JasKiran K Gill, Anna Chatzidaki, Daniel Ursu, Emanuele Sher, Neil S Millar

PLoS One. 2013;8(1):e55047.

PMID: 23383051

1

Expeditious Synthesis, Enantiomeric Resolution, and Enantiomer Functional Characterization of (4-(4-bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): An Allosteric Agonist-Positive Allosteric Modulator of α7 Nicotinic Acetylcholine Receptors

Ganesh A Thakur, Abhijit R Kulkarni, Jeffrey R Deschamps, Roger L Papke

J Med Chem. 2013 Nov 14;56(21):8943-7.

PMID: 24090443

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