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A-803467

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For Research Use Only | Not For Clinical Use
CATAP944261794
CAS944261-79-4
Structure
MDL NumberMFCD10574689
Molecular Weight357.79
InChI KeyVHKBTPQDHDSBSP-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: >10 mg/mL
Assay≥98% (HPLC)
Colorwhite to tan
Formpowder
Size10MG, 50MG
Storage Conditionsroom temp
1

A Selective Nav1.8 Sodium Channel Blocker, A-803467 [5-(4-chlorophenyl-N-(3,5-dimethoxyphenyl)furan-2-carboxamide], Attenuates Spinal Neuronal Activity in Neuropathic Rats

Steve McGaraughty, Katharine L Chu, Marc J C Scanio, Michael E Kort, Connie R Faltynek, Michael F Jarvis

J Pharmacol Exp Ther. 2008 Mar;324(3):1204-11.

PMID: 18089840

1

A-803467, a Potent and Selective Nav1.8 Sodium Channel Blocker, Attenuates Neuropathic and Inflammatory Pain in the Rat

Michael F Jarvis, Prisca Honore, Char-Chang Shieh, Mark Chapman, Shailen Joshi, Xu-Feng Zhang, Michael Kort, William Carroll, Brian Marron, Robert Atkinson, James Thomas, Dong Liu, Michael Krambis, Yi Liu, etc.

Proc Natl Acad Sci U S A. 2007 May 15;104(20):8520-5.

PMID: 17483457

1

A-803467, a Tetrodotoxin-Resistant Sodium Channel Blocker, Modulates ABCG2-mediated MDR in Vitro and in Vivo

Nagaraju Anreddy, Atish Patel, Yun-Kai Zhang, Yi-Jun Wang, Suneet Shukla, Rishil J Kathawala, Priyank Kumar, Pranav Gupta, Suresh V Ambudkar, John N D Wurpel, Zhe-Sheng Chen, Huiqin Guo

Oncotarget. 2015 Nov 17;6(36):39276-91.

PMID: 26515463

1

Absence of Functional Na v 1.8 Channels in Non-diseased Atrial and Ventricular Cardiomyocytes

Simona Casini, Gerard A Marchal, Makiri Kawasaki, Fransisca A Nariswari, Vincent Portero, Nicoline W E van den Berg, Kaomei Guan, Antoine H G Driessen, Marieke W Veldkamp, Isabella Mengarelli, Joris R de Groot, etc.

Cardiovasc Drugs Ther. 2019 Dec;33(6):649-660.

PMID: 31916131

1

The Effects of A-803467 on Cardiac Nav1.5 Channels

Zhonglin Han, Yu Jiang, Feng Xiao, Kejiang Cao, Dao W Wang

Eur J Pharmacol. 2015 May 5;754:52-60.

PMID: 25701724

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