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Col003

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For Research Use Only | Not For Clinical Use
CATAP328565168
CAS328565-16-8
MDL NumberMFCD00852947
Molecular Weight257.24
Description≥98% (HPLC)
SolubilityDMSO: 2 mg/mL, clear
Assay≥98% (HPLC)
Coloryellow to orange
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

A BRET-based Assay Reveals collagen-Hsp47 Interaction Dynamics in the Endoplasmic Reticulum and Small-Molecule Inhibition of This Interaction

Shinya Ito, Masazumi Saito, Masahito Yoshida, Koh Takeuchi, Takayuki Doi, Kazuhiro Nagata

J Biol Chem. 2019 Nov 1;294(44):15962-15972.

PMID: 31492754

1

A Small-Molecule Compound Inhibits a Collagen-Specific Molecular Chaperone and Could Represent a Potential Remedy for Fibrosis

Shinya Ito, Koji Ogawa, Koh Takeuchi, Motoki Takagi, Masahito Yoshida, Takatsugu Hirokawa, Shoshiro Hirayama, Kazuo Shin-Ya, Ichio Shimada, Takayuki Doi, Naoki Goshima, Tohru Natsume, Kazuhiro Nagata

J Biol Chem. 2017 Dec 8;292(49):20076-20085.

PMID: 29025875

1

Structure-Activity Relationship Study on Col-003, a Protein-Protein Interaction Inhibitor Between Collagen and Hsp47

Masahito Yoshida, Masazumi Saito, Shinya Ito, Koji Ogawa, Naoki Goshima, Kazuhiro Nagata, Takayuki Doi

Chem Pharm Bull (Tokyo). 2020 Mar 1;68(3):220-226.

PMID: 31582590

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