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DDR1 Inhibitor 7rh

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For Research Use Only | Not For Clinical Use
CATAP1429617902
CAS1429617-90-2
MDL NumberMFCD30185014
Molecular Weight546.59
Description≥98% (HPLC)
SolubilityDMSO: 10 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

Anticancer Effects of Mesothelin-Targeted Immunotoxin Therapy Are Regulated by Tyrosine Kinase DDR1

Fatima Ali-Rahmani, David J FitzGerald, Scott Martin, Paresma Patel, Marco Prunotto, Pinar Ormanoglu, Craig Thomas, Ira Pastan

Cancer Res. 2016 Mar 15;76(6):1560-8.

PMID: 26719540

1

Antitumor Activity of 7RH, a Discoidin Domain Receptor 1 Inhibitor, Alone or in Combination With Dasatinib Exhibits Antitumor Effects in Nasopharyngeal Carcinoma Cells

Qiu-Ping Lu, Wen-Dan Chen, Jie-Ren Peng, Yao-Dong Xu, Qian Cai, Gong-Kan Feng, Ke Ding, Xiao-Feng Zhu, Zhong Guan

Oncol Lett. 2016 Nov;12(5):3598-3608.

PMID: 27900042

1

Discoidin Domain Receptor 1 Activity Drives an Aggressive Phenotype in Gastric Carcinoma

Hoon Hur, In-Hye Ham, Dakeun Lee, Hyejin Jin, Kristina Y Aguilera, Hye Jeong Oh, Sang-Uk Han, Ji Eun Kwon, Young-Bae Kim, Ke Ding, Rolf A Brekken

BMC Cancer. 2017 Jan 31;17(1):87.

PMID: 28143619

1

Discovery and Optimization of 3-(2-(Pyrazolo[1,5-a]pyrimidin-6-yl)ethynyl)benzamides as Novel Selective and Orally Bioavailable Discoidin Domain Receptor 1 (DDR1) Inhibitors

Mingshan Gao, Lei Duan, Jinfeng Luo, Lianwen Zhang, Xiaoyun Lu, Yan Zhang, Zhang Zhang, Zhengchao Tu, Yong Xu, Xiaomei Ren, Ke Ding

J Med Chem. 2013 Apr 25;56(8):3281-95.

PMID: 23521020

1

Inhibition of Discoidin Domain Receptor 1 Reduces Collagen-mediated Tumorigenicity in Pancreatic Ductal Adenocarcinoma

Kristina Y Aguilera, Huocong Huang, Wenting Du, Moriah M Hagopian, Zhen Wang, Stefan Hinz, Tae Hyun Hwang, Huamin Wang, Jason B Fleming, Diego H Castrillon, Xiaomei Ren, Ke Ding, Rolf A Brekken

Mol Cancer Ther. 2017 Nov;16(11):2473-2485.

PMID: 28864681

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