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Dot1L human

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For Research Use Only | Not For Clinical Use
CATIAR42416071
Descriptionrecombinant, expressed in E. coli, ≥70% (SDS-PAGE)
Assay≥70% (SDS-PAGE)
Formaqueous solution
Size50μG
Storage Conditions−70°C
1

A CRISPR Dropout Screen Identifies Genetic Vulnerabilities and Therapeutic Targets in Acute Myeloid Leukemia

Konstantinos Tzelepis, Hiroko Koike-Yusa, Etienne De Braekeleer, Yilong Li, Emmanouil Metzakopian, Oliver M Dovey, Annalisa Mupo, Vera Grinkevich, Meng Li, Milena Mazan, Malgorzata Gozdecka, Shuhei Ohnishi, etc.

Cell Rep. 2016 Oct 18;17(4):1193-1205.

PMID: 27760321

1

Inhibition of DOT1L and PRMT5 Promote Synergistic Anti-Tumor Activity in a Human MLL Leukemia Model Induced by CRISPR/Cas9

Kathy-Ann Secker, Hildegard Keppeler, Silke Duerr-Stoerzer, Hannes Schmid, Dominik Schneidawind, Thomas Hentrich, Julia M Schulze-Hentrich, Barbara Mankel, Falko Fend, Corina Schneidawind

Oncogene. 2019 Nov;38(46):7181-7195.

PMID: 31417187

1

Structural Basis of Dot1L Stimulation by Histone H2B Lysine 120 Ubiquitination

Marco Igor Valencia-Sánchez, Pablo De Ioannes, Miao Wang, Nikita Vasilyev, Ruoyu Chen, Evgeny Nudler, Jean-Paul Armache, Karim-Jean Armache

Mol Cell. 2019 Jun 6;74(5):1010-1019.e6.

PMID: 30981630

1

The DOT1L Inhibitor Pinometostat Decreases the Host-Response Against Infections: Considerations About Its Use in Human Therapy

Laura Marcos-Villar, Amelia Nieto

Sci Rep. 2019 Nov 14;9(1):16862.

PMID: 31727944

1

The Protective Role of DOT1L in UV-induced Melanomagenesis

Bo Zhu, Shuyang Chen, Hongshen Wang, Chengqian Yin, Changpeng Han, Cong Peng, Zhaoqian Liu, Lixin Wan, Xiaoyang Zhang, Jie Zhang, Christine G Lian, Peilin Ma, Zhi-Xiang Xu, Sharon Prince, Tao Wang, Xiumei Gao, etc.

Nat Commun. 2018 Jan 17;9(1):259.

PMID: 29343685

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