0

EHT 1864

INQUIRY Add to cart
For Research Use Only | Not For Clinical Use
CATAP754240090
CAS754240-09-0
Structure
MDL NumberMFCD11114384
Molecular Weight581.47
InChI KeyLSECOAJFCKFQJG-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityH2O: 10 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size10MG
Storage Conditions2-8°C
1

Characterization of EHT 1864, a Novel Small Molecule Inhibitor of Rac Family Small GTPases

Cercina Onesto, Adam Shutes, Virginie Picard, Fabien Schweighoffer, Channing J Der

Methods Enzymol. 2008;439:111-29.

PMID: 18374160

1

EHT 1864, a Small Molecule Inhibitor of Ras-related C3 Botulinum Toxin Substrate 1 (Rac1), Attenuates Glucose-Stimulated Insulin Secretion in Pancreatic β-cells

Vaibhav Sidarala, Rajakrishnan Veluthakal, Khadija Syeda, Anjaneyulu Kowluru

Cell Signal. 2015 Jun;27(6):1159-67.

PMID: 25725286

1

Rac1 Plays a Role in CXCL12 but Not CCL3-induced Chemotaxis and Rac1 GEF Inhibitor NSC23766 Has Off Target Effects on CXCR4

Shirley C Mills, Lesley Howell, Andrew Beekman, Leanne Stokes, Anja Mueller

Cell Signal. 2018 Jan;42:88-96.

PMID: 29050986

1

Rac-GTPase Promotes Fibrotic TGF-β1 Signaling and Chronic Kidney Disease

Samik Patel, Jiaqi Tang, Jessica M Overstreet, Sandybell Anorga, Fei Lian, Alex Arnouk, Roel Goldschmeding, Paul J Higgins, Rohan Samarakoon

FASEB J. 2019 Sep;33(9):9797-9810.

PMID: 31095421

1

Specificity and Mechanism of Action of EHT 1864, a Novel Small Molecule Inhibitor of Rac Family Small GTPases

Adam Shutes, Cercina Onesto, Virginie Picard, Bertrand Leblond, Fabien Schweighoffer, Channing J Der

J Biol Chem. 2007 Dec 7;282(49):35666-78.

PMID: 17932039

  • Verification code
Contact Us

Send Us a Request

What is your specific need? We will do everything we can to meet your expectations.
Online Inquiry

Online Inquiry

For any inquiry, question or recommendation, please call: or fill out the following form.

  • Verification code

Head Office

  • Tel:
  • Email:

Follow us on

qrcode