CAS 263707-16-0 ESI-09 - Analytical Products / Alfa Chemistry

CAT	AP263707160
CAS	263707-16-0
Molecular Weight	330.77

Description	≥98% (HPLC)
Solubility	DMSO: 20 mg/mL, clear
Assay	≥98% (HPLC)
Color	, faint yellow to dark orange
Form	powder
Size	5MG, 25MG
Storage Conditions	2-8°C

1

Absinthin, an agonist of the bitter taste receptor hTAS2R46, uncovers an ER-to-mitochondria Ca 2+-shuttling event

Maria Talmon, Silvia Rossi, Dmitry Lim, Federica Pollastro, Gioele Palattella, Federico A Ruffinatti, Patrizia Marotta, Renzo Boldorini, Armando A Genazzani, Luigia G Fresu

J Biol Chem. 2019 Aug 16;294(33):12472-12482.

PMID: 31248983

1

Biochemical and Pharmacological Characterizations of ESI-09 Based EPAC Inhibitors: Defining the ESI-09 "Therapeutic Window"

Yingmin Zhu, Haijun Chen, Stephen Boulton, Fang Mei, Na Ye, Giuseppe Melacini, Jia Zhou, Xiaodong Cheng

Sci Rep. 2015 Mar 20;5:9344.

PMID: 25791905

1

Efficient Synthesis of ESI-09, A Novel Non-cyclic Nucleotide EPAC Antagonist

Haijun Chen, Chunyong Ding, Christopher Wild, Huiling Liu, Tianzhi Wang, Mark A White, Xiaodong Cheng, Jia Zhou

Tetrahedron Lett. 2013 Mar 20;54(12):1546-1549.

PMID: 23459418

1

Exchange Protein Directly Activated by cAMP (Epac) Protects Against Airway Inflammation and Airway Remodeling in Asthmatic Mice

Yi-Fei Chen, Ge Huang, Yi-Min Wang, Ming Cheng, Fang-Fang Zhu, Jin-Nan Zhong, Ya-Dong Gao

Respir Res. 2019 Dec 18;20(1):285.

PMID: 31852500

1

Lithium and an EPAC-specific Inhibitor ESI-09 Synergistically Suppress Pancreatic Cancer Cell Proliferation and Survival

Xinshuo Wang, Cheng Luo, Xiaodong Cheng, Meiling Lu

Acta Biochim Biophys Sin (Shanghai). 2017 Jul 1;49(7):573-580.

PMID: 28475672

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