CAS 337972-47-1 FAUC 213 - Analytical Products / Alfa Chemistry

CAT	AP337972471
CAS	337972-47-1
Structure
MDL Number	MFCD06798338
Molecular Weight	326.82
InChI Key	DTRXURJDKOYCCD-UHFFFAOYSA-N

Description	≥98% (HPLC), solid
Solubility	DMSO: ~24 mg/mL (with warming up to 60 °C); H2O: insoluble
Assay	≥98% (HPLC)
Color	white
Form	solid
Size	5MG, 25MG
Storage Conditions	2-8°C

1

Blocking alpha2A Adrenoceptors, but Not Dopamine Receptors, Augments Bupropion-Induced Hypophagia in Rats

Sanna K Janhunen, Susanne E la Fleur, Roger A H Adan

Obesity (Silver Spring). 2013 Dec;21(12):E700-8.

PMID: 23894096

1

FAUC 213, a Highly Selective Dopamine D4 Receptor Full Antagonist, Exhibits Atypical Antipsychotic Properties in Behavioural and Neurochemical Models of Schizophrenia

Frank Boeckler, Holger Russig, Weining Zhang, Stefan Löber, John Schetz, Harald Hübner, Boris Ferger, Peter Gmeiner, Joram Feldon

Psychopharmacology (Berl). 2004 Aug;175(1):7-17.

PMID: 15007532

1

Rationally Based Efficacy Tuning of Selective Dopamine d4 Receptor Ligands Leading to the Complete Antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213)

S Löber, H Hübner, W Utz, P Gmeiner

J Med Chem. 2001 Aug 16;44(17):2691-4.

PMID: 11495580

1

Synthesis, Radiofluorination, and in Vitro Evaluation of pyrazolo[1,5-a]pyridine-based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET

Olaf Prante, Rainer Tietze, Carsten Hocke, Stefan Löber, Harald Hübner, Torsten Kuwert, Peter Gmeiner

J Med Chem. 2008 Mar 27;51(6):1800-10.

PMID: 18307287

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