GSK2801

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For Research Use Only | Not For Clinical Use

CAT	IAR4246389
MDL Number	MFCD26142953
Molecular Weight	371.45
InChI Key	KHWCPNJRJCNVRI-UHFFFAOYSA-N

Description	≥98% (HPLC)
Solubility	DMSO: 10 mg/mL, clear
Assay	≥98% (HPLC)
Color	, white to pink to light brown
Form	powder
Size	5MG, 25MG
Storage Conditions	−20°C

Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B

Peiling Chen, Apirat Chaikuad, Paul Bamborough, Marcus Bantscheff, Chas Bountra, Chun-Wa Chung, Oleg Fedorov, Paola Grandi, David Jung, Robert Lesniak, Matthew Lindon, Susanne Müller, Martin Philpott, Rab Prinjha, etc.

J Med Chem. 2016 Feb 25;59(4):1410-24.

PMID: 25799074

GSK2801, a BAZ2/BRD9 Bromodomain Inhibitor, Synergizes With BET Inhibitors to Induce Apoptosis in Triple-Negative Breast Cancer

Samantha M Bevill, Jose F Olivares-Quintero, Noah Sciaky, Brian T Golitz, Darshan Singh, Adriana S Beltran, Naim U Rashid, Timothy J Stuhlmiller, Andrew Hale, Nathaniel J Moorman, Charlene M Santos, Steven P Angus, etc.

Mol Cancer Res. 2019 Jul;17(7):1503-1518.

PMID: 31000582

Hepatitis Delta Virus Histone Mimicry Drives the Recruitment of Chromatin Remodelers for Viral RNA Replication

Natali Abeywickrama-Samarakoon, Jean-Claude Cortay, Camille Sureau, Susanne Müller, Dulce Alfaiate, Francesca Guerrieri, Apirat Chaikuad, Martin Schröder, Philippe Merle, Massimo Levrero, Paul Dény

Nat Commun. 2020 Jan 21;11(1):419.

PMID: 31964889

Recognition of hyperacetylated N-terminus of H2AZ by TbBDF2 from Trypanosoma brucei

Xiao Yang, Xuelei Wu, Jiahai Zhang, Xuecheng Zhang, Chao Xu, Shanhui Liao, Xiaoming Tu

Biochem J. 2017 Nov 9;474(22):3817-3830.

PMID: 29025975

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