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IU1

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For Research Use Only | Not For Clinical Use
CATAP314245335
CAS314245-33-5
Structure
MDL NumberMFCD01917473
Molecular Weight300.37
InChI KeyJUWDSDKJBMFLHE-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: >10 mg/mL
Assay≥98% (HPLC)
Coloroff-white to light brown
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

An Inhibitor of the Proteasomal Deubiquitinating Enzyme USP14 Induces Tau Elimination in Cultured Neurons

Monica Boselli, Byung-Hoon Lee, Jessica Robert, Miguel A Prado, Sang-Won Min, Chialin Cheng, M Catarina Silva, Changhyun Seong, Suzanne Elsasser, Ketki M Hatle, Timothy C Gahman, Steven P Gygi, Stephen J Haggarty, etc.

J Biol Chem. 2017 Nov 24;292(47):19209-19225.

PMID: 28972160

1

Inhibition of USP14 Enhances the Sensitivity of Breast Cancer to Enzalutamide

Xiaohong Xia, Chuyi Huang, Yuning Liao, Yuan Liu, Jinchan He, Zhiqiang Guo, Lili Jiang, Xuejun Wang, Jinbao Liu, Hongbiao Huang

J Exp Clin Cancer Res. 2019 May 24;38(1):220.

PMID: 31126320

1

M2 Microglia-Derived Exosomes Protect the Mouse Brain From Ischemia-Reperfusion Injury via Exosomal miR-124

Yaying Song, Zongwei Li, Tingting He, Meijie Qu, Lu Jiang, Wanlu Li, Xiaojing Shi, Jiaji Pan, Linyuan Zhang, Yongting Wang, Zhijun Zhang, Yaohui Tang, Guo-Yuan Yang

Theranostics. 2019 May 4;9(10):2910-2923.

PMID: 31244932

1

Neurotoxic Mechanisms by Which the USP14 Inhibitor IU1 Depletes Ubiquitinated Proteins and Tau in Rat Cerebral Cortical Neurons: Relevance to Alzheimer's Disease

Magdalena J Kiprowska, Anna Stepanova, Dustin R Todaro, Alexander Galkin, Arthur Haas, Scott M Wilson, Maria E Figueiredo-Pereira

Biochim Biophys Acta Mol Basis Dis. 2017 Jun;1863(6):1157-1170.

PMID: 28372990

1

Small Molecule Inhibitors Reveal Allosteric Regulation of USP14 via Steric Blockade

Yiwei Wang, Yuxuan Jiang, Shan Ding, Jiawang Li, Ningjing Song, Yujing Ren, Danning Hong, Cai Wu, Bin Li, Feng Wang, Wei He, Jiawei Wang, Ziqing Mei

Cell Res. 2018 Dec;28(12):1186-1194.

PMID: 30254335

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