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JNJ-47965567

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For Research Use Only | Not For Clinical Use
CATAP1428327314
CAS1428327-31-4
MDL NumberMFCD28334214
Molecular Weight488.64
Description≥98% (HPLC)
SolubilityDMSO: 20 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

Critical Evaluation of P2X7 Receptor Antagonists in Selected Seizure Models

Wolfgang Fischer, Heike Franke, Ute Krügel, Heiko Müller, Klaus Dinkel, Brian Lord, Michael A Letavic, David C Henshall, Tobias Engel

PLoS One. 2016 Jun 9;11(6):e0156468.

PMID: 27281030

1

Pharmacological Characterization of a Novel Centrally Permeable P2X7 Receptor Antagonist: JNJ-47965567

Anindya Bhattacharya, Qi Wang, Hong Ao, James R Shoblock, Brian Lord, Leah Aluisio, Ian Fraser, Diane Nepomuceno, Robert A Neff, Natalie Welty, Timothy W Lovenberg, Pascal Bonaventure, Alan D Wickenden, etc.

Br J Pharmacol. 2013 Oct;170(3):624-40.

PMID: 23889535

1

The P2X7 Receptor Antagonist JNJ-47965567 Administered Thrice Weekly From Disease Onset Does Not Alter Progression of Amyotrophic Lateral Sclerosis in SOD1

Diane Ly, Anjila Dongol, Peter Cuthbertson, Thomas V Guy, Nicholas J Geraghty, Reece A Sophocleous, Lucia Sin, Bradley J Turner, Debbie Watson, Justin J Yerbury, Ronald Sluyter

Purinergic Signal. 2020 Mar;16(1):109-122.

PMID: 32170537

1

The Role of P2X7 Receptors in a Rodent PCP-induced Schizophrenia Model

Bence Koványi, Cecilia Csölle, Stefano Calovi, Adrienn Hanuska, Erzsébet Kató, László Köles, Anindya Bhattacharya, József Haller, Beáta Sperlágh

Sci Rep. 2016 Nov 8;6:36680.

PMID: 27824163

1

Transient P2X7 Receptor Antagonism Produces Lasting Reductions in Spontaneous Seizures and Gliosis in Experimental Temporal Lobe Epilepsy

Alba Jimenez-Pacheco, Miguel Diaz-Hernandez, Marina Arribas-Blázquez, Amaya Sanz-Rodriguez, Luis A Olivos-Oré, Antonio R Artalejo, Mariana Alves, Michael Letavic, M Teresa Miras-Portugal, Ronan M Conroy, etc.

J Neurosci. 2016 Jun 1;36(22):5920-32.

PMID: 27251615

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