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KRN633

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For Research Use Only | Not For Clinical Use
CATAP286370158
CAS286370-15-8
Structure
Molecular Weight416.86
Description≥98% (HPLC)
SolubilityDMSO: 3 mg/mL, clear (warmed)
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions−20°C
1

Attenuation of Retinal Endothelial Vasodilator Function in a Rat Model of Retinopathy of Prematurity

Ayuki Nakano, Asami Mori, Shiho Arima, Daiki Asano, Akane Morita, Kenji Sakamoto, Tohru Nagamitsu, Tsutomu Nakahara

Curr Eye Res. 2019 Dec;44(12):1360-1368.

PMID: 31317786

1

KRN633, an Inhibitor of Vascular Endothelial Growth Factor Receptor Tyrosine Kinase, Induces Intrauterine Growth Restriction in Mice

Naomichi Abe, Tsutomu Nakahara, Akane Morita, Yoshiko Wada, Asami Mori, Kenji Sakamoto, Tohru Nagamitsu, Kunio Ishii

Birth Defects Res B Dev Reprod Toxicol. 2013 Aug;98(4):297-303.

PMID: 23780833

1

KRN633: A Selective Inhibitor of Vascular Endothelial Growth Factor receptor-2 Tyrosine Kinase That Suppresses Tumor Angiogenesis and Growth

Kazuhide Nakamura, Atsushi Yamamoto, Masaru Kamishohara, Kazumi Takahashi, Eri Taguchi, Toru Miura, Kazuo Kubo, Masabumi Shibuya, Toshiyuki Isoe

Mol Cancer Ther. 2004 Dec;3(12):1639-49.

PMID: 15634658

1

Platelet-Rich Plasma Prevents In Vitro Transforming Growth Factor-β1-Induced Fibroblast to Myofibroblast Transition: Involvement of Vascular Endothelial Growth Factor (VEGF)-A/VEGF Receptor-1-Mediated Signaling

Flaminia Chellini, Alessia Tani, Larissa Vallone, Daniele Nosi, Paola Pavan, Franco Bambi, Sandra Zecchi Orlandini, Chiara Sassoli

Cells. 2018 Sep 19;7(9):142.

PMID: 30235859

1

Short-term Treatment With VEGF Receptor Inhibitors Induces Retinopathy of Prematurity-Like Abnormal Vascular Growth in Neonatal Rats

Ayuki Nakano, Tsutomu Nakahara, Asami Mori, Hiroko Ushikubo, Kenji Sakamoto, Kunio Ishii

Exp Eye Res. 2016 Feb;143:120-31.

PMID: 26500193

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