0

LDN-214117

INQUIRY Add to cart
For Research Use Only | Not For Clinical Use
CATIAR4243898
Molecular Weight419.52
InChI KeyBHUXVRVMMYAXKN-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: 10 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

ALK2 inhibitors display beneficial effects in preclinical models of ACVR1 mutant diffuse intrinsic pontine glioma

Diana Carvalho, Kathryn R Taylor, Nagore Gene Olaciregui, Valeria Molinari, Matthew Clarke, Alan Mackay, Ruth Ruddle, Alan Henley, Melanie Valenti, Angela Hayes, Alexis De Haven Brandon, Suzanne A Eccles, etc.

Commun Biol. 2019 May 9;2:156.

PMID: 31098401

1

Inhibition of Bone Morphogenetic Protein Signaling Reduces Viability, Growth and Migratory Potential of Non-Small Cell Lung Carcinoma Cells

Jelena Mihajlović, Laura A M Diehl, Andreas Hochhaus, Joachim H Clement

J Cancer Res Clin Oncol. 2019 Nov;145(11):2675-2687.

PMID: 31531741

1

Pharmacologic Strategies for Assaying BMP Signaling Function

Teresa Dinter, Geoffrey A Bocobo, Paul B Yu

Methods Mol Biol. 2019;1891:221-233.

PMID: 30414136

1

Structure-activity Relationship of 3,5-diaryl-2-aminopyridine ALK2 Inhibitors Reveals Unaltered Binding Affinity for Fibrodysplasia Ossificans Progressiva Causing Mutants

Agustin H Mohedas, You Wang, Caroline E Sanvitale, Peter Canning, Sungwoon Choi, Xuechao Xing, Alex N Bullock, Gregory D Cuny, Paul B Yu

J Med Chem. 2014 Oct 9;57(19):7900-15.

PMID: 25101911

1

Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma

Deeba Ensan, David Smil, Carlos A Zepeda-Velázquez, Dimitrios Panagopoulos, Jong Fu Wong, Eleanor P Williams, Roslin Adamson, Alex N Bullock, Taira Kiyota, Ahmed Aman, Owen G Roberts, Aled M Edwards, Jeff A O'Meara, etc.

J Med Chem. 2020 May 14;63(9):4978-4996.

PMID: 32369358

  • Verification code
Contact Us

Send Us a Request

What is your specific need? We will do everything we can to meet your expectations.
Online Inquiry

Online Inquiry

For any inquiry, question or recommendation, please call: or fill out the following form.

  • Verification code

Head Office

  • Tel:
  • Email:

Follow us on

qrcode