CAS 333962-91-7 LUF5834 - Analytical Products / Alfa Chemistry

CAT	AP333962917
CAS	333962-91-7
Structure
Molecular Weight	348.38

Description	≥98% (HPLC)
Solubility	DMSO: 20 mg/mL, clear
Assay	≥98% (HPLC)
Color	white to beige
Form	powder
Size	5MG, 25MG
Storage Conditions	−20°C

1

A Novel Nonribose Agonist, LUF5834, Engages Residues That Are Distinct From Those of Adenosine-Like Ligands to Activate the Adenosine A(2a) Receptor

J Robert Lane, Carmen Klein Herenbrink, Gerard J P van Westen, Jelle A Spoorendonk, Carsten Hoffmann, Adriaan P IJzerman

Mol Pharmacol. 2012 Mar;81(3):475-87.

PMID: 22188926

1

Activation of the A2A Adenosine G-protein-coupled Receptor by Conformational Selection

Libin Ye, Ned Van Eps, Marco Zimmer, Oliver P Ernst, R Scott Prosser

Nature. 2016 May 12;533(7602):265-8.

PMID: 27144352

1

Characterization of [3H]LUF5834: A Novel Non-Ribose High-Affinity Agonist Radioligand for the Adenosine A1 Receptor

J Robert Lane, Elisabeth Klaasse, Judy Lin, John van Bruchem, Margot W Beukers, Adriaan P Ijzerman

Biochem Pharmacol. 2010 Oct 15;80(8):1180-9.

PMID: 20599769

1

New, Non-Adenosine, High-Potency Agonists for the Human Adenosine A2B Receptor With an Improved Selectivity Profile Compared to the Reference Agonist N-ethylcarboxamidoadenosine

Margot W Beukers, Lisa C W Chang, Jacobien K von Frijtag Drabbe Künzel, Thea Mulder-Krieger, Ronald F Spanjersberg, Johannes Brussee, Ad P IJzerman

J Med Chem. 2004 Jul 15;47(15):3707-9.

PMID: 15239649

1

Validation of a Na +-shift binding assay for estimation of the intrinsic efficacy of ligands at the A 2A adenosine receptor

François Noël, Fernando M do Monte

J Pharmacol Toxicol Methods. Mar-Apr 2017;84:51-56.

PMID: 27810394

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