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P5091

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For Research Use Only | Not For Clinical Use
CATAP882257116
CAS882257-11-6
Molecular Weight348.22
Description≥98% (HPLC)
SolubilityDMSO: 10 mg/mL, clear
Assay≥98% (HPLC)
Colorlight yellow to dark yellow
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

A Small Molecule Inhibitor of Ubiquitin-Specific protease-7 Induces Apoptosis in Multiple Myeloma Cells and Overcomes Bortezomib Resistance

Dharminder Chauhan, Ze Tian, Benjamin Nicholson, K G Suresh Kumar, Bin Zhou, Ruben Carrasco, Jeffrey L McDermott, Craig A Leach, Mariaterresa Fulcinniti, Matthew P Kodrasov, Joseph Weinstock, William D Kingsbury, etc.

Cancer Cell. 2012 Sep 11;22(3):345-58.

PMID: 22975377

1

CCDC6 and USP7 Expression Levels Suggest Novel Treatment Options in High-Grade Urothelial Bladder Cancer

Francesco Morra, Francesco Merolla, Daniela Criscuolo, Luigi Insabato, Riccardo Giannella, Gennaro Ilardi, Aniello Cerrato, Roberta Visconti, Stefania Staibano, Angela Celetti

J Exp Clin Cancer Res. 2019 Feb 20;38(1):90.

PMID: 30786932

1

Genome-scale CRISPR-Cas9 screen identifies druggable dependencies in TP53 wild-type Ewing sarcoma

Björn Stolte, Amanda Balboni Iniguez, Neekesh V Dharia, Amanda L Robichaud, Amy Saur Conway, Ann M Morgan, Gabriela Alexe, Nathan J Schauer, Xiaoxi Liu, Gregory H Bird, Aviad Tsherniak, Francisca Vazquez, etc.

J Exp Med. 2018 Aug 6;215(8):2137-2155.

PMID: 30045945

1

Pharmacological Inhibition of USP7 Promotes Antitumor Immunity and Contributes to Colon Cancer Therapy

Changqing Fu, Xiaojue Zhu, Peiqi Xu, Yonghao Li

Onco Targets Ther. 2019 Jan 15;12:609-617.

PMID: 30697058

1

The Combined Effect of USP7 Inhibitors and PARP Inhibitors in Hormone-Sensitive and Castration-Resistant Prostate Cancer Cells

Francesco Morra, Francesco Merolla, Virginia Napolitano, Gennaro Ilardi, Caterina Miro, Simona Paladino, Stefania Staibano, Aniello Cerrato, Angela Celetti

Oncotarget. 2017 May 9;8(19):31815-31829.

PMID: 28415632

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