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PDE7A active rat

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For Research Use Only | Not For Clinical Use
CATIAR4245724
Descriptionrecombinant, expressed in baculovirus infected Sf9 cells, ≥30% (SDS-PAGE)
Assay≥30% (SDS-PAGE)
Formaqueous solution
Size10μG
Storage Conditions−70°C
1

Expression and Regulation of Cyclic Nucleotide Phosphodiesterases in Human and Rat Pancreatic Islets

Emilia Heimann, Helena A Jones, Svante Resjö, Vincent C Manganiello, Lena Stenson, Eva Degerman

PLoS One. 2010 Dec 1;5(12):e14191.

PMID: 21152070

1

Modulation of cAMP-specific PDE Without Emetogenic Activity: New Sulfide-Like PDE7 Inhibitors

Ana M García, José Brea, Jose A Morales-García, Daniel I Perez, Alejandro González, Sandra Alonso-Gil, Irene Gracia-Rubio, Clara Ros-Simó, Santiago Conde, María Isabel Cadavid, María Isabel Loza, Ana Perez-Castillo, etc.

J Med Chem. 2014 Oct 23;57(20):8590-607.

PMID: 25264825

1

Novel Amide Derivatives of 1,3-dimethyl-2,6-dioxopurin-7-yl-alkylcarboxylic Acids as Multifunctional TRPA1 Antagonists and PDE4/7 Inhibitors: A New Approach for the Treatment of Pain

Grażyna Chłoń-Rzepa, Marietta Ślusarczyk, Agnieszka Jankowska, Alicja Gawalska, Adam Bucki, Marcin Kołaczkowski, Artur Świerczek, Krzysztof Pociecha, Elżbieta Wyska, Małgorzata Zygmunt, Grzegorz Kazek, etc.

Eur J Med Chem. 2018 Oct 5;158:517-533.

PMID: 30245393

1

Novel Butanehydrazide Derivatives of purine-2,6-dione as Dual PDE4/7 Inhibitors With Potential Anti-Inflammatory Activity: Design, Synthesis and Biological Evaluation

Grażyna Chłoń-Rzepa, Agnieszka Jankowska, Marietta Ślusarczyk, Artur Świerczek, Krzysztof Pociecha, Elżbieta Wyska, Adam Bucki, Alicja Gawalska, Marcin Kołaczkowski, Maciej Pawłowski

Eur J Med Chem. 2018 Feb 25;146:381-394.

PMID: 29407965

1

The SAR Development of Dihydroimidazoisoquinoline Derivatives as Phosphodiesterase 10A Inhibitors for the Treatment of Schizophrenia

Ginny D Ho, W Michael Seganish, Ana Bercovici, Deen Tulshian, William J Greenlee, Rachel Van Rijn, Alan Hruza, Li Xiao, Diane Rindgen, Deborra Mullins, Mario Guzzi, Xiaoping Zhang, Carina Bleickardt, Robert Hodgson

Bioorg Med Chem Lett. 2012 Apr 1;22(7):2585-9.

PMID: 22377514

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