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PF-477736

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For Research Use Only | Not For Clinical Use
CATAP952021602
CAS952021-60-2
MDL NumberMFCD16038847
Molecular Weight419.48
InChI KeyNDEXUOWTGYUVGA-LJQANCHMSA-N
Description≥98% (HPLC)
SolubilityDMSO: ≥20 mg/mL
Assay≥98% (HPLC)
Coloryellow
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

Co-Inhibition of the DNA Damage Response and CHK1 Enhances Apoptosis of Neuroblastoma Cells

Kiyohiro Ando, Yohko Nakamura, Hiroki Nagase, Akira Nakagawara, Tsugumichi Koshinaga, Satoshi Wada, Makoto Makishima

Int J Mol Sci. 2019 Jul 29;20(15):3700.

PMID: 31362335

1

DUOXA1-mediated ROS Production Promotes Cisplatin Resistance by Activating ATR-Chk1 Pathway in Ovarian Cancer

Yunxiao Meng, Chi-Wei Chen, Mingo M H Yung, Wei Sun, Jing Sun, Zhuqing Li, Jing Li, Zongzhu Li, Wei Zhou, Stephanie S Liu, Annie N Y Cheung, Hextan Y S Ngan, John C Braisted, Yan Kai, Weiqun Peng, Alexandros Tzatsos, etc.

Cancer Lett. 2018 Aug 1;428:104-116.

PMID: 29704517

1

Gemcitabine and CHK1 Inhibition Potentiate EGFR-directed Radioimmunotherapy Against Pancreatic Ductal Adenocarcinoma

Fares Al-Ejeh, Marina Pajic, Wei Shi, Murugan Kalimutho, Mariska Miranda, Adnan M Nagrial, Angela Chou, Andrew V Biankin, Sean M Grimmond, Australian Pancreatic Cancer Genome Initiative, Michael P Brown, etc.

Clin Cancer Res. 2014 Jun 15;20(12):3187-97.

PMID: 24838526

1

Lessons From LIMK1 Enzymology and Their Impact on Inhibitor Design

Eidarus Salah, Deep Chatterjee, Alessandra Beltrami, Anthony Tumber, Franziska Preuss, Peter Canning, Apirat Chaikuad, Petra Knaus, Stefan Knapp, Alex N Bullock, Sebastian Mathea

Biochem J. 2019 Nov 15;476(21):3197-3209.

PMID: 31652302

1

Thymineless Death by the Fluoropyrimidine Polymer F10 Involves Replication Fork Collapse and Is Enhanced by Chk1 Inhibition

Chinnadurai Mani, Sachin Pai, Cinta Maria Papke, Komaraiah Palle, William H Gmeiner

Neoplasia. 2018 Dec;20(12):1236-1245.

PMID: 30439567

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