0

Phosphodiesterase 5A1 human

INQUIRY Add to cart
For Research Use Only | Not For Clinical Use
CATIAR42415175
Descriptionrecombinant, expressed in Sf9 cells
Size10μG
Storage Conditions−70°C
1

A Multi-Biochemical and In Silico Study on Anti-Enzymatic Actions of Pyroglutamic Acid Against PDE-5, ACE, and Urease Using Various Analytical Techniques: Unexplored Pharmacological Properties and Cytotoxicity Evaluation

Miroslava Šudomová, Sherif T S Hassan, Haroon Khan, Mahsa Rasekhian, Seyed Mohammad Nabavi

Biomolecules. 2019 Aug 21;9(9):392.

PMID: 31438631

1

Cyclic Nucleotide Phosphodiesterase Type 4 Inhibitors: Evaluation of pyrazolo[1,5-a]-1,3,5-triazine Ring System as an Adenine Bioisostere

Pierre Raboisson, Dominique Schultz, Christian Muller, Jean-Marie Reimund, Guillaume Pinna, Romain Mathieu, Philippe Bernard, Quoc-Tuan Do, Renee L Desjarlais, Hélène Justiano, Claire Lugnier, Jean-Jacques Bourguignon

Eur J Med Chem. 2008 Apr;43(4):816-29.

PMID: 17640774

1

High Biochemical Selectivity of Tadalafil, Sildenafil and Vardenafil for Human Phosphodiesterase 5A1 (PDE5) Over PDE11A4 Suggests the Absence of PDE11A4 Cross-Reaction in Patients

J L Weeks, R Zoraghi, A Beasley, K R Sekhar, S H Francis, J D Corbin

Int J Impot Res. Jan-Feb 2005;17(1):5-9.

PMID: 15538396

1

Phosphodiesterase-5 Isoforms: Differential Cyclic Guanyl Monophosphate Binding and Cyclic Guanyl Monophosphate Catalytic Activities, and Inhibitory Effects of Sildenafil and Vardenafil

Guiting Lin, Zhong-Cheng Xin, Tom F Lue, Ching-Shwun Lin

J Urol. 2006 Sep;176(3):1242-7.

PMID: 16890733

1

Potent Inhibition of Human phosphodiesterase-5 by Icariin Derivatives

Mario Dell'Agli, Germana V Galli, Esther Dal Cero, Federica Belluti, Riccardo Matera, Elisa Zironi, Giampiero Pagliuca, Enrica Bosisio

J Nat Prod. 2008 Sep;71(9):1513-7.

PMID: 18778098

  • Verification code
Contact Us

Send Us a Request

What is your specific need? We will do everything we can to meet your expectations.
Online Inquiry

Online Inquiry

For any inquiry, question or recommendation, please call: or fill out the following form.

  • Verification code

Head Office

  • Tel:
  • Email:

Follow us on

qrcode