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PRMT4 Active human

INQUIRY Add to cart
For Research Use Only | Not For Clinical Use
CATIAR42416084
Descriptionrecombinant, expressed in baculovirus infected insect cells, ≥65% (SDS-PAGE)
Assay≥65% (SDS-PAGE)
Formaqueous solution
Size20μG
Storage Conditions−70°C
1

Hijacking DNA Methyltransferase Transition State Analogues to Produce Chemical Scaffolds for PRMT Inhibitors

Ludovic Halby, Nils Marechal, Dany Pechalrieu, Vincent Cura, Don-Marc Franchini, Céline Faux, Fréderic Alby, Nathalie Troffer-Charlier, Srikanth Kudithipudi, Albert Jeltsch, Wahiba Aouadi, Etienne Decroly, etc.

Philos Trans R Soc Lond B Biol Sci. 2018 Jun 5;373(1748):20170072.

PMID: 29685976

1

TP-064, a Potent and Selective Small Molecule Inhibitor of PRMT4 for Multiple Myeloma

Kazuhide Nakayama, Magdalena M Szewczyk, Carlo Dela Sena, Hong Wu, Aiping Dong, Hong Zeng, Fengling Li, Renato Ferreira de Freitas, Mohammad S Eram, Matthieu Schapira, Yuji Baba, Mihoko Kunitomo, Douglas R Cary, etc.

Oncotarget. 2018 Apr 6;9(26):18480-18493.

PMID: 29719619

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