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RQ-00203078

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For Research Use Only | Not For Clinical Use
CATAP1254205521
CAS1254205-52-1
MDL NumberMFCD29049510
Molecular Weight554.85
InChI KeyIJGQFZYYEHCCIZ-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: 25 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

Effects of Menthol and Its Interaction With Nicotine-Conditioned Cue on Nicotine-Seeking Behavior in Rats

Erin Harrison, Lisa Biswas, Ramachandram Avusula, Meiyu Zhang, Yongzhen Gong, Xiu Liu

Psychopharmacology (Berl). 2017 Dec;234(23-24):3443-3453.

PMID: 28918457

1

Functional Role of the Transient Receptor Potential Melastatin 8 (TRPM8) Ion Channel in the Urinary Bladder Assessed by Conscious Cystometry and Ex Vivo Measurements of Single-Unit Mechanosensitive Bladder Afferent Activities in the Rat

Hiroki Ito, Naoki Aizawa, Rino Sugiyama, Shuzo Watanabe, Nobuyuki Takahashi, Masaomi Tajimi, Hiroshi Fukuhara, Yukio Homma, Yoshinobu Kubota, Karl-Erik Andersson, Yasuhiko Igawa

BJU Int. 2016 Mar;117(3):484-94.

PMID: 26189966

1

Identification of a Novel 2-pyridyl-benzensulfonamide Derivative, RQ-00203078, as a Selective and Orally Active TRPM8 Antagonist

Masashi Ohmi, Yuji Shishido, Tadashi Inoue, Kazuo Ando, Akiyoshi Fujiuchi, Akiko Yamada, Shuzo Watanabe, Kiyoshi Kawamura

Bioorg Med Chem Lett. 2014 Dec 1;24(23):5364-8.

PMID: 25455182

1

Pharmacological Inhibition of TRPM8-induced Gene Transcription

Gerald Thiel, Tobias M Backes, Jennifer Welck, Sebastian Steinhausen, Anna-Lena Fischer, Daniel S Langfermann, Myriam Ulrich, Ulrich Wissenbach, Oliver G Rössler

Biochem Pharmacol. 2019 Dec;170:113678.

PMID: 31654626

1

The Transient Receptor Potential Vanilloid 4 Agonist RN-1747 Inhibits the Calcium Response to Histamine

Beatrix Pfanzagl, Roswitha Pfragner, Erika Jensen-Jarolim

Pharmacology. 2019;104(3-4):166-172.

PMID: 31212298

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