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S1P4 Receptor Antagonist, CYM50358

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For Research Use Only | Not For Clinical Use
CATIAR42414760
Molecular Weight389.28
DescriptionThe S1P4 Receptor Antagonist, CYM50358 controls the biological activity of S1P4 Receptor. This small molecule/inhibitor is primarily used for Biochemicals applications.
SolubilityDMSO: 100 mg/mL, clear, colorless
Assay≥98% (HPLC)
Colorwhite
Formsolid; protect from light
Size5MG
Storage Conditions+2C to +8C
1

Blockade of Sphingosine 1-Phosphate Receptor 2 Signaling Attenuates High-Fat Diet-Induced Adipocyte Hypertrophy and Systemic Glucose Intolerance in Mice

Yoshihiko Kitada, Kazuo Kajita, Koichiro Taguchi, Ichiro Mori, Masahiro Yamauchi, Takahide Ikeda, Mikako Kawashima, Motochika Asano, Toshiko Kajita, Tatsuo Ishizuka, Yoshiko Banno, Itaru Kojima, Jerold Chun, etc.

Endocrinology. 2016 May;157(5):1839-51.

PMID: 26943364

1

Sphingosine 1-phosphate (S1P) Suppresses the Collagen-Induced Activation of Human Platelets via S1P4 Receptor

Takashi Onuma, Kumiko Tanabe, Yuko Kito, Masanori Tsujimoto, Kodai Uematsu, Yukiko Enomoto, Rie Matsushima-Nishiwaki, Tomoaki Doi, Kiyoshi Nagase, Shigeru Akamatsu, Haruhiko Tokuda, Shinji Ogura, Toru Iwama, etc.

Thromb Res. 2017 Aug;156:91-100.

PMID: 28609704

1

TGFβ1 Evokes Myoblast Apoptotic Response via a Novel Signaling Pathway Involving S1P4 Transactivation Upstream of Rho-kinase-2 Activation

Francesca Cencetti, Caterina Bernacchioni, Francesca Tonelli, Edward Roberts, Chiara Donati, Paola Bruni

FASEB J. 2013 Nov;27(11):4532-46.

PMID: 23913862

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