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SAK3

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For Research Use Only | Not For Clinical Use
CATAP1256269870
CAS1256269-87-0
Molecular Weight369.41
Description≥98% (HPLC)
SolubilityDMSO: 2 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

Pharmacological properties of SAK3, a novel T-type voltage-gated Ca 2+ channel enhancer

Yasushi Yabuki, Kazuya Matsuo, Hisanao Izumi, Hidaka Haga, Takashi Yoshida, Minoru Wakamori, Akikazu Kakei, Kenji Sakimura, Takaichi Fukuda, Kohji Fukunaga

Neuropharmacology. 2017 May 1;117:1-13.

PMID: 28093211

1

SAK3-Induced Neuroprotection Is Mediated by Nicotinic Acetylcholine Receptors

Kohji Fukunaga, Yasushi Yabuki, Akinori Akaike, Shun Shimohama, Yoshimi Misu

PMID: 31314408

1

The Disease-modifying Drug Candidate, SAK3 Improves Cognitive Impairment and Inhibits Amyloid Beta Deposition in App Knock-in Mice

Hisanao Izumi, Yasuharu Shinoda, Takashi Saito, Takaomi C Saido, Keita Sato, Yasushi Yabuki, Yotaro Matsumoto, Yoshitomi Kanemitsu, Yoshihisa Tomioka, Nona Abolhassani, Yusaku Nakabeppu, Kohji Fukunaga

Neuroscience. 2018 May 1;377:87-97.

PMID: 29510211

1

T-type Calcium Channel Enhancer SAK3 Produces Anti-Depressant-Like Effects by Promoting Adult Hippocampal Neurogenesis in Olfactory Bulbectomized Mice

Jing Xu, Yasushi Yabuki, Mengze Yu, Kohji Fukunaga

J Pharmacol Sci. 2018 Aug;137(4):333-341.

PMID: 30196018

1

T-type Calcium Channel Enhancer SAK3 Promotes Dopamine and Serotonin Releases in the Hippocampus in Naive and Amyloid Precursor Protein Knock-In Mice

Shuo Wang, Yasushi Yabuki, Kazuya Matsuo, Jing Xu, Hisanao Izumi, Kenji Sakimura, Takashi Saito, Takaomi C Saido, Kohji Fukunaga

PLoS One. 2018 Dec 20;13(12):e0206986.

PMID: 30571684

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