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SirReal2

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For Research Use Only | Not For Clinical Use
CATAP709002460
CAS709002-46-0
Molecular Weight420.55
InChI KeyMENNDDDTIIZDDN-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: 20 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions−20°C
1

Direct Comparison of SIRT2 Inhibitors: Potency, Specificity, Activity-Dependent Inhibition, and On-Target Anticancer Activities

Nicole A Spiegelman, Ian R Price, Hui Jing, Miao Wang, Min Yang, Ji Cao, Jun Young Hong, Xiaoyu Zhang, Pornpun Aramsangtienchai, Sushabhan Sadhukhan, Hening Lin

ChemMedChem. 2018 Sep 19;13(18):1890-1894.

PMID: 30058233

1

SIRT2 Functions in Aging, Autophagy, and Apoptosis in Post-Maturation Bovine Oocytes

Dejun Xu, Xiaohan Jiang, Huanshan He, Dingbang Liu, Li Yang, Huali Chen, Lin Wu, Guoxia Geng, Qingwang Li

Life Sci. 2019 Sep 1;232:116639.

PMID: 31295472

1

SIRT2 Inhibition Results in Meiotic Arrest, Mitochondrial Dysfunction, and Disturbance of Redox Homeostasis During Bovine Oocyte Maturation

Dejun Xu, Lin Wu, Xiaohan Jiang, Li Yang, Jianyong Cheng, Huali Chen, Rongmao Hua, Guoxia Geng, Lulu Yang, Qingwang Li

Int J Mol Sci. 2019 Mar 18;20(6):1365.

PMID: 30889926

1

SIRT2 Plays a Novel Role on Progesterone, Estradiol and Testosterone Synthesis via PPARs/LXRα Pathways in Bovine Ovarian Granular Cells

Dejun Xu, Huanshan He, Xiaohan Jiang, Rongmao Hua, Huali Chen, Li Yang, Jianyong Cheng, Jiaxin Duan, Qingwang Li

J Steroid Biochem Mol Biol. 2019 Jan;185:27-38.

PMID: 30009951

1

SIRT2 Promotes the Migration and Invasion of Gastric Cancer Through RAS/ERK/JNK/MMP-9 Pathway by Increasing PEPCK1-Related Metabolism

Yang Li, Mingming Zhang, Robert G Dorfman, Yida Pan, Dehua Tang, Lei Xu, Zhenguo Zhao, Qian Zhou, Lixing Zhou, Yuming Wang, Yuyao Yin, Shanshan Shen, Bo Kong, Helmut Friess, Shimin Zhao, Lei Wang, Xiaoping Zou

Neoplasia. 2018 Jul;20(7):745-756.

PMID: 29925042

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