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SK-216

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For Research Use Only | Not For Clinical Use
CATAP654080032
CAS654080-03-2
Molecular Weight533.52
Description≥98% (HPLC)
SolubilityH2O: 0.5 mg/mL, clear (warmed)
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditionsroom temp
1

Inhibition of PAI-1 Limits Tumor Angiogenesis Regardless of Angiogenic Stimuli in Malignant Pleural Mesothelioma

Yusuke Takayama, Noboru Hattori, Hironobu Hamada, Takeshi Masuda, Keitaro Omori, Shin Akita, Hiroshi Iwamoto, Kazunori Fujitaka, Nobuoki Kohno

Cancer Res. 2016 Jun 1;76(11):3285-94.

PMID: 27197170

1

Inhibition of Plasminogen Activator Inhibitor-1 Attenuates Transforming Growth Factor-β-Dependent Epithelial Mesenchymal Transition and Differentiation of Fibroblasts to Myofibroblasts

Keitaro Omori, Noboru Hattori, Tadashi Senoo, Yusuke Takayama, Takeshi Masuda, Taku Nakashima, Hiroshi Iwamoto, Kazunori Fujitaka, Hironobu Hamada, Nobuoki Kohno

PLoS One. 2016 Feb 9;11(2):e0148969.

PMID: 26859294

1

Plasminogen Activator inhibitor-1 (Pai-1) Blockers Suppress Intestinal Polyp Formation in Min Mice

Michihiro Mutoh, Naoko Niho, Masami Komiya, Mami Takahashi, Rina Ohtsubo, Kiyoshi Nakatogawa, Kentaro Ueda, Takashi Sugimura, Keiji Wakabayashi

Carcinogenesis. 2008 Apr;29(4):824-9.

PMID: 18258607

1

SK-216, a Novel Inhibitor of Plasminogen Activator Inhibitor-1, Suppresses Lung Metastasis of Human Osteosarcoma

Minori Tsuge, Mitsuhiko Osaki, Ryo Sasaki, Mio Hirahata, Futoshi Okada

Int J Mol Sci. 2018 Mar 5;19(3):736.

PMID: 29510576

1

SK-216, an Inhibitor of Plasminogen Activator inhibitor-1, Limits Tumor Progression and Angiogenesis

Takeshi Masuda, Noboru Hattori, Tadashi Senoo, Shin Akita, Nobuhisa Ishikawa, Kazunori Fujitaka, Yoshinori Haruta, Hiroshi Murai, Nobuoki Kohno

Mol Cancer Ther. 2013 Nov;12(11):2378-88.

PMID: 23990114

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