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SKLB1002

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For Research Use Only | Not For Clinical Use
CATAP1225451842
CAS1225451-84-2
MDL NumberMFCD27938707
Molecular Weight320.39
InChI KeyRQVGFDBMONQTBC-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: 2 mg/mL, clear (warmed)
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

A New Selective Vascular Endothelial Growth Factor Receptor 2 Inhibitor Ablates Disease in a Mouse Model of Psoriasis

Heng-Xiu Yan, Yong Wang, Xiao-Nong Yang, Li-Xin Fu, Dong-Mei Tang

Mol Med Rep. 2013 Aug;8(2):434-8.

PMID: 23732650

1

SKLB1002, a Novel Inhibitor of VEGF Receptor 2 Signaling, Induces Vascular Normalization to Improve Systemically Administered Chemotherapy Efficacy

G Shen, Y Li, T Du, G Shi, L Dai, X Chen, R Zheng, W Li, X Su, S Zhang, Y Wei, S Yang, H Deng

Neoplasma. 2012;59(5):486-93.

PMID: 22668017

1

SKLB1002, a Novel Potent Inhibitor of VEGF Receptor 2 Signaling, Inhibits Angiogenesis and Tumor Growth in Vivo

Shuang Zhang, Zhixing Cao, Hongwei Tian, Guobo Shen, Yongping Ma, Huanzhang Xie, Yalin Liu, Chengjian Zhao, Senyi Deng, Yang Yang, Renlin Zheng, Weiwei Li, Na Zhang, Shengyong Liu, Wei Wang, Lixia Dai, etc.

Clin Cancer Res. 2011 Jul 1;17(13):4439-50.

PMID: 21622720

1

Synergic Antitumor Effect of SKLB1002 and Local Hyperthermia in 4T1 and CT26

Wen Nie, Xue-lei Ma, Ya-xiong Sang, Yu-li Li, Xiang Gao, Guang-chao Xu, Guo-bo Shen, Hua-shan Shi, Xiao-xiao Liu, Feng-tian Wang, Yu-quan Wei

Clin Exp Med. 2014 May;14(2):203-13.

PMID: 23263406

1

VEGFR2 Regulates Endothelial Differentiation of Colon Cancer Cells

Zhiyong Liu, Lisha Qi, Yixian Li, Xiulan Zhao, Baocun Sun

BMC Cancer. 2017 Aug 30;17(1):593.

PMID: 28854900

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