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Spautin-1

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For Research Use Only | Not For Clinical Use
CATAP1262888287
CAS1262888-28-7
Structure
MDL NumberMFCD16962292
Molecular Weight271.26
InChI KeyAWIVHRPYFSSVOG-UHFFFAOYSA-N
Description≥98% (HPLC)
SolubilityDMSO: 15 mg/mL (clear solution)
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditions2-8°C
1

Beclin1 Controls the Levels of p53 by Regulating the Deubiquitination Activity of USP10 and USP13

Junli Liu, Hongguang Xia, Minsu Kim, Lihua Xu, Ying Li, Lihong Zhang, Yu Cai, Helin Vakifahmetoglu Norberg, Tao Zhang, Tsuyoshi Furuya, Minzhi Jin, Zhimin Zhu, Huanchen Wang, Jia Yu, Yanxia Li, Yan Hao, etc.

Cell. 2011 Sep 30;147(1):223-34.

PMID: 21962518

1

Inhibition of EGFR Signaling With Spautin-1 Represents a Novel Therapeutics for Prostate Cancer

Yuning Liao, Zhiqiang Guo, Xiaohong Xia, Yuan Liu, Chuyi Huang, Lili Jiang, Xuejun Wang, Jinbao Liu, Hongbiao Huang

J Exp Clin Cancer Res. 2019 Apr 11;38(1):157.

PMID: 30975171

1

Spautin-1 Ameliorates Acute Pancreatitis via Inhibiting Impaired Autophagy and Alleviating Calcium Overload

Juan Xiao, Xueping Feng, Xiao-Ying Huang, Zhongshi Huang, Yanqiang Huang, Chaogan Li, Genliang Li, Song Nong, Ruoshi Wu, Yongzhi Huang, Xi-Dai Long

Mol Med. 2016 Oct;22:643-652.

PMID: 27579473

1

Spautin-1, a Novel Autophagy Inhibitor, Enhances Imatinib-Induced Apoptosis in Chronic Myeloid Leukemia

Shan Shao, Su Li, Youwen Qin, Xiaorui Wang, Yining Yang, Haitao Bai, Lili Zhou, Chuxian Zhao, Chun Wang

Int J Oncol. 2014 May;44(5):1661-8.

PMID: 24585095

1

The Autophagy Inhibitor Spautin-1 Antagonizes Rescue of Mutant CFTR Through an Autophagy-Independent and USP13-Mediated Mechanism

Emanuela Pesce, Elvira Sondo, Loretta Ferrera, Valeria Tomati, Emanuela Caci, Paolo Scudieri, Ilaria Musante, Mario Renda, Nesrine Baatallah, Nathalie Servel, Alexandre Hinzpeter, Diego di Bernardo, Nicoletta Pedemonte, etc.

Front Pharmacol. 2018 Dec 13;9:1464.

PMID: 30618756

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