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Tesaglitazar

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For Research Use Only | Not For Clinical Use
CATAP251565852
CAS251565-85-2
Structure
MDL NumberMFCD07784004
Molecular Weight408.47
InChI KeyCXGTZJYQWSUFET-IBGZPJMESA-N
Description≥98% (HPLC)
SolubilityDMSO: 20 mg/mL, clear
Assay≥98% (HPLC)
Colorwhite to beige
Formpowder
Size5MG, 25MG
Storage Conditionsroom temp
1

Dual peroxisome-proliferator-activated-receptor-α/γ Activation Inhibits SIRT1-PGC1α Axis and Causes Cardiac Dysfunction

Charikleia Kalliora, Ioannis D Kyriazis, Shin-Ichi Oka, Melissa J Lieu, Yujia Yue, Estela Area-Gomez, Christine J Pol, Ying Tian, Wataru Mizushima, Adave Chin, Diego Scerbo, P Christian Schulze, Mete Civelek, etc.

JCI Insight. 2019 Aug 8;5(17):e129556.

PMID: 31393858

1

Effects of Dual Peroxisome Proliferator-Activated Receptors

Mohammad Alsalem, Mansour Haddad, Sara A Aldossary, Heba Kalbouneh, Belal Azab, Aala Dweik, Amer Imraish, Khalid El-Salem

PPAR Res. 2019 Apr 17;2019:2630232.

PMID: 31139213

1

Tesaglitazar

Niklaus Kamber, Timothy M E Davis

IDrugs. 2005 Nov;8(11):927-35.

PMID: 16254788

1

Tesaglitazar Ameliorates Non-Alcoholic Fatty Liver Disease and Atherosclerosis Development in Diabetic Low-Density Lipoprotein Receptor-Deficient Mice

Bu-Chun Zhang, Wei-Ming Li, Xian-Kai Li, Meng-Yun Zhu, Wen-Liang Che, Ya-Wei Xu

Exp Ther Med. 2012 Dec;4(6):987-992.

PMID: 23226761

1

Tesaglitazar, a Novel Dual Peroxisome Proliferator-Activated Receptor alpha/gamma Agonist, Dose-Dependently Improves the Metabolic Abnormalities Associated With Insulin Resistance in a Non-Diabetic Population

B Fagerberg, S Edwards, T Halmos, J Lopatynski, H Schuster, S Stender, G Stoa-Birketvedt, S Tonstad, S Halldórsdóttir, I Gause-Nilsson

Diabetologia. 2005 Sep;48(9):1716-25.

PMID: 16001233

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