CAS 1229591-56-3 UCPH-102 - Analytical Products / Alfa Chemistry

CAT	AP1229591563
CAS	1229591-56-3
Molecular Weight	330.38

Description	≥98% (HPLC)
Solubility	DMSO: 20 mg/mL, clear
Assay	≥98% (HPLC)
Color	white to beige
Form	powder
Size	5MG, 25MG
Storage Conditions	2-8°C

1

Allosteric Modulation of an Excitatory Amino Acid Transporter: The Subtype-Selective Inhibitor UCPH-101 Exerts Sustained Inhibition of EAAT1 Through an Intramonomeric Site in the Trimerization Domain

Bjarke Abrahamsen, Nicole Schneider, Mette N Erichsen, Tri H V Huynh, Christoph Fahlke, Lennart Bunch, Anders A Jensen

J Neurosci. 2013 Jan 16;33(3):1068-87.

PMID: 23325245

1

Bioavailability Studies and in Vitro Profiling of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor UCPH-102

Isabell Haym, Tri H V Huynh, Stinne W Hansen, Martin H F Pedersen, Josep A Ruiz, Mette N Erichsen, Mikko Gynther, Walden E Bjørn-Yoshimoto, Bjarke Abrahamsen, Jesper F Bastlund, Christoffer Bundgaard, Anette L Eriksen, etc.

ChemMedChem. 2016 Feb 17;11(4):403-19.

PMID: 26797816

1

Design, Synthesis and Pharmacological Characterization of Coumarin-Based Fluorescent Analogs of Excitatory Amino Acid Transporter Subtype 1 Selective Inhibitors, UCPH-101 and UCPH-102

Tri H V Huynh, Bjarke Abrahamsen, Karsten K Madsen, Alba Gonzalez-Franquesa, Anders A Jensen, Lennart Bunch

Bioorg Med Chem. 2012 Dec 1;20(23):6831-9.

PMID: 23072958

1

New Insight Into the Structure-Activity Relationships of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors UCPH-101 and UCPH-102

Stinne W Hansen, Mette N Erichsen, Tri H V Huynh, Josep A Ruiz, Isabell Haym, Walden E Bjørn-Yoshimoto, Bjarke Abrahamsen, Jeanette Hansen, Morten Storgaard, Anette L Eriksen, Anders A Jensen, Lennart Bunch

ChemMedChem. 2016 Feb 17;11(4):382-402.

PMID: 26757239

1

Probing for Improved Potency and in Vivo Bioavailability of Excitatory Amino Acid Transporter Subtype 1 Inhibitors UCPH-101 and UCPH-102: Design, Synthesis and Pharmacological Evaluation of Substituted 7-biphenyl Analogs

Mette N Erichsen, Jeanette Hansen, Josep A Ruiz, Charles S Demmer, Bjarke Abrahamsen, Jesper F Bastlund, Christoffer Bundgaard, Anders A Jensen, Lennart Bunch

Neurochem Res. 2014 Oct;39(10):1964-79.

PMID: 24682739

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