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WP1130

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For Research Use Only | Not For Clinical Use
CATIAR42410931
Molecular Weight384.27
DescriptionA cell-permeable tyrphostin compound that acts as a partially selective deubiquitinase (DUB) inhibitor and suppresses JAK-Stat signaling pathway.
SolubilityDMSO: 100 mg/mL
Assay≥97% (HPLC)
Colorlight yellow
Formsolid; protect from light
Size10MG
Storage Conditions+2C to +8C
1

Deubiquitinase Inhibition by Small-Molecule WP1130 Triggers Aggresome Formation and Tumor Cell Apoptosis

Vaibhav Kapuria, Luke F Peterson, Dexing Fang, William G Bornmann, Moshe Talpaz, Nicholas J Donato

Cancer Res. 2010 Nov 15;70(22):9265-76.

PMID: 21045142

1

Dub3 Inhibition Suppresses Breast Cancer Invasion and Metastasis by Promoting Snail1 Degradation

Yadi Wu, Yu Wang, Yiwei Lin, Yajuan Liu, Yifan Wang, Jianhang Jia, Puja Singh, Young-In Chi, Chi Wang, Chenfang Dong, Wei Li, Min Tao, Dana Napier, Qiuying Shi, Jiong Deng, B Mark Evers, Binhua P Zhou

Nat Commun. 2017 Feb 15;8:14228.

PMID: 28198361

1

Inhibition of USP9X Induces Apoptosis in FLT3-ITD-positive AML Cells Cooperatively by Inhibiting the Mutant Kinase Through Aggresomal Translocation and Inducing Oxidative Stress

Hiroki Akiyama, Yoshihiro Umezawa, Shinya Ishida, Keigo Okada, Ayako Nogami, Osamu Miura

Cancer Lett. 2019 Jul 1;453:84-94.

PMID: 30946869

1

USP9X Inhibition Improves Gemcitabine Sensitivity in Pancreatic Cancer by Inhibiting Autophagy

Tao Ma, Wei Chen, Xiao Zhi, Hao Liu, Yue Zhou, Brayant Wei Chen, Liqiang Hu, Jian Shen, Xiaoxiao Zheng, Shufen Zhang, Bo Zhang, Haijun Li, Tingbo Liang

Cancer Lett. 2018 Nov 1;436:129-138.

PMID: 30118840

1

WP1130 Enhances TRAIL-Induced Apoptosis Through USP9X-Dependent miR-708-Mediated Downregulation of c-FLIP

Seok Kim, Seon Min Woo, Kyoung-Jin Min, Seung Un Seo, Tae-Jin Lee, Peter Kubatka, Dong Eun Kim, Taeg Kyu Kwon

Cancers (Basel). 2019 Mar 11;11(3):344.

PMID: 30862047

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